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A-68930 hydrochloride

CAS No. 130465-39-3

A-68930 hydrochloride ( A68930 )

产品货号. M11221 CAS No. 130465-39-3

A-68930 is a potent, specific, orally bioavailable agonist of the D1 Dopamine receptor with EC50 of 2.5 nM.

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥2219 有现货
50MG ¥8068 有现货
100MG ¥12798 有现货
200MG 获取报价 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    A-68930 hydrochloride
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    A-68930 is a potent, specific, orally bioavailable agonist of the D1 Dopamine receptor with EC50 of 2.5 nM.
  • 产品描述
    A-68930 is a potent, specific, orally bioavailable agonist of the D1 Dopamine receptor with EC50 of 2.5 nM; shows a much weaker agonist (EC50=3,920 nM) at the D2 dopamine receptor; demonstrates antidepressant and anorectic effects in animal models without stimulant effects.Heart Failure Discontinued
  • 同义词
    A68930
  • 通路
    GPCR/G Protein
  • 靶点
    Dopamine Receptor
  • 受体
    Dopamine Receptor
  • 研究领域
    Neurological Disease
  • 适应症
    ——

化学信息

  • CAS Number
    130465-39-3
  • 分子量
    307.77
  • 分子式
    C16H17NO3 · HCl
  • 纯度
    >98% (HPLC)
  • 溶解度
    ——
  • SMILES
    C1C(OC(C2=C1C(=C(C=C2)O)O)CN)C3=CC=CC=C3.Cl
  • 化学全称
    1H-2-Benzopyran-5,6-diol, 1-(aminomethyl)-3,4-dihydro-3-phenyl-, hydrochloride, (1R,3S)-rel- (9CI)

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1. Kebabian JW, et al. Am J Hypertens. 1990 Jun;3(6 Pt 2):40S-42S.
2. Trampus M, et al. Eur J Pharmacol. 1993 Apr 22;235(1):83-7.
3. AI-Naser HA, et al. Behav Pharmacol. 1994 Apr;5(2):210-218.
产品手册
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